nitroimidazoles xi [i]. syntheses of disubstituted nitroimidazolylquinolines
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reaction of substituted-aniline (8) with ethyl (l-methyl-5-nitroimidazole-2- carbonyl) acetate (9) gave 4-hydroxy-2-(l-methyl-5-nitro-2-imidazolyl)- substituted-quinolines (lo), which were converted to compound 11 with phosphorus oxychloride. substituted-2-(l-methyl-5-nitro-2-imidazo1yl)-4.- methyl-(or phenyl-) quinolines (14) were prepared through the reaction of 2- acetyl-5-nitro-1-methyl-imidazole (13) with 0-aminoacetophenones (or oaminobenzophenones) in acid medium
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Journal title:
journal of sciences islamic republic of iranجلد ۶، شماره ۱، صفحات ۰-۰
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